Amazi meza ya Lidocaine Hydrochloride 73-78-9 Utanga Lidocaine Hcl uturuka mubushinwa
Ibikoresho bya Shimi & Umubiri
Izina Rusange | Lidocaine hydrochloride | ||
---|---|---|---|
Numero ya CAS | 73-78-9 | Uburemere bwa molekile | 270.798 |
Ubucucike | N / A. | Ingingo yo guteka | 350.8ºC kuri 760 mmHg |
Inzira ya molekulari | C14H23ClN2O | Ingingo yo gushonga | 80-82 ° C. |
MSDS | N / A. | Flash Flash | 166ºC |
Gukoresha hydrochloride ya LidocaineLidocaine Hclumunyu, amide anesthetic yaho, ifite imiti igabanya ubukana muri vitro no muri vivo, bishoboka ko biterwa no kwiyongera kwa cytokine ya pro-inflammatory, molekules ya adhesion-1 (ICAM-1), no kugabanya neutrophile yinjira.Intego: Lidocaine ni imiti isanzwe ya anesthetic na antarrhythmic.Lidocaine ikoreshwa cyane cyane kugirango igabanye kwandura, gutwikwa no kubabara biturutse ku gutwika uruhu, guterwa nk'inyo yo kuvura amenyo cyangwa nka anestheque yaho yo kubaga bito.Lidocaine, amine yambere ya amide-ubwoko bwa anesthetic yaho, yashizwemo bwa mbere mwizina rya xylocaine numu chimiste wo muri Suwede Nils Lofgren mumwaka wa 1943. Mugenzi we Bengt Lundqvist yakoze ubushakashatsi bwa mbere bwo gutera inshinge kuri we.Lidocaine igera kuri 95% metabolised (dealkylated) muri. umwijima na CYP3A4 kuri farumasi ikora ya metabolite monoethylglycinexylidide (MEGX) hanyuma ikagera kuri glycine idakora.MEGX ifite ubuzima burebure burenze lidocaine ariko kandi ni umuyoboro muke wa sodiumi.Kurandura igice cya kabiri cya lidocaine ni iminota 90-120 kubarwayi benshi.Ibi birashobora kumara igihe kinini kubarwayi bafite ubumuga bwumwijima (impuzandengo yiminota 343) cyangwa kunanirwa k'umutima (impuzandengo yiminota 136). |
Aliase: LIDOCAINE HCL, Xyloneural, Xilina hydrochloride, Lidocaton, Xylocard
Isuku: 99%
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Ibibazo:
Q1: Nshobora kubona ingero zimwe?
Igisubizo: Yego, turashobora gutanga icyitegererezo cyubusa, ariko igiciro cyo kohereza cyishyurwa nabakiriya bacu.
Q2: Nigute ushobora gutangira ibicuruzwa cyangwa kwishyura?
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Q3: Nigute ushobora kwemeza ubuziranenge bwibicuruzwa mbere yo gutanga amabwiriza?
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Q4: MOQ yawe ni iki?
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